English

• 

• 1. [1] J.E. Biggs-Houck, A. Younai, J.T. Shaw, Recent advances in multicomponent reactions for diversity-oriented synthesis, Curr. Opin. Chem. Biol. 14 (2010) 371-382.[1] J.E. Biggs-Houck, A. Younai, J.T. Shaw, Recent advances in multicomponent reactions for diversity-oriented synthesis, Curr. Opin. Chem. Biol. 14 (2010) 371-382.

  2. [2] B.B. Touré, D.G. Hall, Natural product synthesis using multicomponent reaction strategies, Chem. Rev. 109 (2009) 4439-4486.[2] B.B. Touré, D.G. Hall, Natural product synthesis using multicomponent reaction strategies, Chem. Rev. 109 (2009) 4439-4486.

  3. [3] J.Y. Lu, X.Y. Gong, H.J. Yang, H. Fu, Concise copper-catalyzed one-pot tandem synthesis of benzimidazo[1,2-b]isoquinolin-11-one derivatives, Chem. Commun. 46 (2010) 4172-4174.[3] J.Y. Lu, X.Y. Gong, H.J. Yang, H. Fu, Concise copper-catalyzed one-pot tandem synthesis of benzimidazo[1,2-b]isoquinolin-11-one derivatives, Chem. Commun. 46 (2010) 4172-4174.

  4. [4] Y.G. Zhu, C.W. Zhai, Y.L. Yue, L.P. Yang, W.H. Hu, One-pot three-component tandem reaction of diazo compounds with anilines and unsaturated ketoesters: a novel synthesis of 2,3-dihydropyrrole derivatives, Chem. Commun. 11 (2009) 1362-1364.[4] Y.G. Zhu, C.W. Zhai, Y.L. Yue, L.P. Yang, W.H. Hu, One-pot three-component tandem reaction of diazo compounds with anilines and unsaturated ketoesters: a novel synthesis of 2,3-dihydropyrrole derivatives, Chem. Commun. 11 (2009) 1362-1364.

  5. [5] B. Ganem, Strategies for innovation in multicomponent reaction design, Acc. Chem. Res. 42 (2009) 463-472.[5] B. Ganem, Strategies for innovation in multicomponent reaction design, Acc. Chem. Res. 42 (2009) 463-472.

  6. [6] H. Bienayme, C. Hulme, G. Oddon, P. Schmitt, Maximizing synthetic efficiency: multi-component transformations lead the way, Chem. Eur. J. 6 (2000) 3321- 3329.[6] H. Bienayme, C. Hulme, G. Oddon, P. Schmitt, Maximizing synthetic efficiency: multi-component transformations lead the way, Chem. Eur. J. 6 (2000) 3321- 3329.

  7. [7] A. Domling, I. Ugi, Multicomponent reactions with isocyanides, Angew. Chem. Int. Ed. 39 (2000) 3168-3210.[7] A. Domling, I. Ugi, Multicomponent reactions with isocyanides, Angew. Chem. Int. Ed. 39 (2000) 3168-3210.

  8. [8] J.P. Zhu, Recent developments in the isonitrile-based multicomponent synthesis of heterocycles, Eur. J. Org. Chem. 7 (2003) 1133-1144.[8] J.P. Zhu, Recent developments in the isonitrile-based multicomponent synthesis of heterocycles, Eur. J. Org. Chem. 7 (2003) 1133-1144.

  9. [9] D.J. Ramon, M. Yus, Asymmetric multicomponent reactions (AMCRs): the new frontier, Angew. Chem. Int. Ed. 44 (2005) 1602-1634.[9] D.J. Ramon, M. Yus, Asymmetric multicomponent reactions (AMCRs): the new frontier, Angew. Chem. Int. Ed. 44 (2005) 1602-1634.

  10. [10] W.T. Ashton, L.L. Chang, K.L. Flanagan, et al., Triazolinone biphenylsulfonamide derivatives as orally active angiotensin Ⅱ antagonists with potent AT1 receptor affinity and enhanced AT2 affinity, J. Med. Chem. 37 (1994) 2808-2824.[10] W.T. Ashton, L.L. Chang, K.L. Flanagan, et al., Triazolinone biphenylsulfonamide derivatives as orally active angiotensin Ⅱ antagonists with potent AT1 receptor affinity and enhanced AT2 affinity, J. Med. Chem. 37 (1994) 2808-2824.

  11. [11] N. Demirbas, A. Demirbas, S.A. Karaoglu, Synthesis and biological activities of new 1,2,4-triazole-3-one derivatives, Russ. J. Bioorg. Chem. 31 (2005) 387-397.[11] N. Demirbas, A. Demirbas, S.A. Karaoglu, Synthesis and biological activities of new 1,2,4-triazole-3-one derivatives, Russ. J. Bioorg. Chem. 31 (2005) 387-397.

  12. [12] N. Demirbasş, R. Ugurluoglu, A. Demirbasş, Synthesis of 3-alkyl(aryl)-4-alkylidenamino- 4,5-dihydro-1H-1,2,4-triazol-5-ones and 3-alkyl-4-alkylamino-4,5- dihydro-1H-1,2,4-triazol-5-ones as antitumor agents, Bioorg. Med. Chem. 10 (2002) 3717-3723.[12] N. Demirbasş, R. Ugurluoglu, A. Demirbasş, Synthesis of 3-alkyl(aryl)-4-alkylidenamino- 4,5-dihydro-1H-1,2,4-triazol-5-ones and 3-alkyl-4-alkylamino-4,5- dihydro-1H-1,2,4-triazol-5-ones as antitumor agents, Bioorg. Med. Chem. 10 (2002) 3717-3723.

  13. [13] N.S. Khalil, Efficient synthesis of novel 1,2,4-triazole fused acyclic and 21-28 membered macrocyclic and/or lariat macrocyclic oxaazathia crown compounds with potential antimicrobial activity, Eur. J. Med. Chem. 45 (2010) 5265-5277.[13] N.S. Khalil, Efficient synthesis of novel 1,2,4-triazole fused acyclic and 21-28 membered macrocyclic and/or lariat macrocyclic oxaazathia crown compounds with potential antimicrobial activity, Eur. J. Med. Chem. 45 (2010) 5265-5277.

  14. [14] J.M. Kane, B.M. Baron, M.W. Dudley, et al., 2,4-Dihydro-3H-1,2,4-triazol-3-ones as anticonvulsant agents, J. Med. Chem. 33 (1990) 2772-2777.[14] J.M. Kane, B.M. Baron, M.W. Dudley, et al., 2,4-Dihydro-3H-1,2,4-triazol-3-ones as anticonvulsant agents, J. Med. Chem. 33 (1990) 2772-2777.

  15. [15] C.Q. Shen, X.Y. Che, W.Y. Wang, et al., Design and synthesis of novel triazole antifungal derivatives by structure-based bioisosterism, Eur. J. Med. Chem. 46 (2011) 5276-5282.[15] C.Q. Shen, X.Y. Che, W.Y. Wang, et al., Design and synthesis of novel triazole antifungal derivatives by structure-based bioisosterism, Eur. J. Med. Chem. 46 (2011) 5276-5282.

  16. [16] G. Aperis, E. Mylonakis, Newer triazole antifungal agents: pharmacology, spectrum, clinical efficacy and limitations, Expert Opin. Investig. Drugs 15 (2006) 579- 602.[16] G. Aperis, E. Mylonakis, Newer triazole antifungal agents: pharmacology, spectrum, clinical efficacy and limitations, Expert Opin. Investig. Drugs 15 (2006) 579- 602.

  17. [17] A. Davoodnia, M. Bakavoli, M. Soleimany, H. Behmadi, A new one-pot neat synthesis of 1,2,4-triazol-3-ones through 4-(N,N-dimethylamino) pyridine (DMAP) catalyzed cyclocondensation of ethyl carbazate with aryl nitriles, Chin. Chem. Lett. 19 (2008) 685-688.[17] A. Davoodnia, M. Bakavoli, M. Soleimany, H. Behmadi, A new one-pot neat synthesis of 1,2,4-triazol-3-ones through 4-(N,N-dimethylamino) pyridine (DMAP) catalyzed cyclocondensation of ethyl carbazate with aryl nitriles, Chin. Chem. Lett. 19 (2008) 685-688.

  18. [18] H. Gadegoni, S. Manda, Synthesis and screening of some novel substituted indoles contained 1,3,4-oxadiazole and 1,2,4-triazole moiety, Chin. Chem. Lett. 24 (2013) 127-130.[18] H. Gadegoni, S. Manda, Synthesis and screening of some novel substituted indoles contained 1,3,4-oxadiazole and 1,2,4-triazole moiety, Chin. Chem. Lett. 24 (2013) 127-130.

  19. [19] H. Tang, C. Zheng, X. Ren, et al., Synthesis and biological evaluation of novel triazole derivatives as antifungal agents, Chin. Chem. Lett. 24 (2013) 219-222.[19] H. Tang, C. Zheng, X. Ren, et al., Synthesis and biological evaluation of novel triazole derivatives as antifungal agents, Chin. Chem. Lett. 24 (2013) 219-222.

  20. [20] P.Z. Zhang, S.F. Zhou, T.R. Li, L. Jiang, Efficient synthesis and in vitro antifungal activity of 1H-benzimidazol-1-yl acetates/propionates containing 1H-1,2,4-triazole moiety, Chin. Chem. Lett. 23 (2012) 1381-1384.[20] P.Z. Zhang, S.F. Zhou, T.R. Li, L. Jiang, Efficient synthesis and in vitro antifungal activity of 1H-benzimidazol-1-yl acetates/propionates containing 1H-1,2,4-triazole moiety, Chin. Chem. Lett. 23 (2012) 1381-1384.

  21. [21] X. Qin, H.B. Yu, H. Dai, et al., Synthesis and plant-growth regulatory activities of novel imine derivatives containing 1H-1,2,4-triazole and thiazole rings, Chin. Chem. Lett. 21 (2010) 283-286.[21] X. Qin, H.B. Yu, H. Dai, et al., Synthesis and plant-growth regulatory activities of novel imine derivatives containing 1H-1,2,4-triazole and thiazole rings, Chin. Chem. Lett. 21 (2010) 283-286.

  22. [22] J.R. Kavaji, O. Kotresh, B.V. Badami, Chemical reactivity of 3-aryl-5-methyl-1,3,4- oxadiazolin-2-ones towards nitrogen nucleophiles, J. Chem. Res. (2003) 275-278.[22] J.R. Kavaji, O. Kotresh, B.V. Badami, Chemical reactivity of 3-aryl-5-methyl-1,3,4- oxadiazolin-2-ones towards nitrogen nucleophiles, J. Chem. Res. (2003) 275-278.

  23. [23] I. Kawasaki, A. Domen, S. Kataoka, et al., A new synthetic method for substituted 2,4-dihydro-3H-1,2,4-triazol-3-ones and 3-thiones via 1,4-dialkyl-5-phenylthio- 1H-1,2,4-triazolium salts, Heterocycles 60 (2003) 351-363.[23] I. Kawasaki, A. Domen, S. Kataoka, et al., A new synthetic method for substituted 2,4-dihydro-3H-1,2,4-triazol-3-ones and 3-thiones via 1,4-dialkyl-5-phenylthio- 1H-1,2,4-triazolium salts, Heterocycles 60 (2003) 351-363.

  24. [24] J.Z. Deng, C.S. Burgey, A novel and efficient synthesis of 2,5-substituted 1,2,4- triazol-3-ones, Tetrahedron Lett. 46 (2005) 7993-7996.[24] J.Z. Deng, C.S. Burgey, A novel and efficient synthesis of 2,5-substituted 1,2,4- triazol-3-ones, Tetrahedron Lett. 46 (2005) 7993-7996.

  25. [25] H. Chouaieb, M. Ben Mosbah, M. Kossentini, M. Salem, Novel method for the synthesis of 1,2,4-triazoles and 1,2,4-triazol-3-ones, Synth. Commun. 33 (2003) 3861-3868.[25] H. Chouaieb, M. Ben Mosbah, M. Kossentini, M. Salem, Novel method for the synthesis of 1,2,4-triazoles and 1,2,4-triazol-3-ones, Synth. Commun. 33 (2003) 3861-3868.

  26. [26] S. Kamiya, K. Yamaguchi, M. Miyahara, N. Miyata, Cyclization of 1-aryl-1-nitroso- 3-(2-pyridylmethyl)ureas to1-aryl-5-(2-pyridyl)-2,4-dihydro-1,2,4-triazolo-3- ones, Chem. Pharm. Bull. 38 (1990) 3226-3229.[26] S. Kamiya, K. Yamaguchi, M. Miyahara, N. Miyata, Cyclization of 1-aryl-1-nitroso- 3-(2-pyridylmethyl)ureas to1-aryl-5-(2-pyridyl)-2,4-dihydro-1,2,4-triazolo-3- ones, Chem. Pharm. Bull. 38 (1990) 3226-3229.

  27. [27] M. Chen, X.F. Wang, S.S. Wang, et al., Synthesis, characterization and fungicidal activities of novel fluorinated 3,5-disubstituted-4H-1,2,4-triazol-4-amines, J. Fluor. Chem. 135 (2012) 323-329.[27] M. Chen, X.F. Wang, S.S. Wang, et al., Synthesis, characterization and fungicidal activities of novel fluorinated 3,5-disubstituted-4H-1,2,4-triazol-4-amines, J. Fluor. Chem. 135 (2012) 323-329.

  28. [28] S.R. Devineni, S. Doddaga, R. Donka, N.R. Chamarthi, CeCl₃·7H2O-SiO2: catalyst promoted microwave assisted neat synthesis, antifungal and antioxidant activities of a-diaminophosphonates, Chin. Chem. Lett. 24 (2013) 759-763.[28] S.R. Devineni, S. Doddaga, R. Donka, N.R. Chamarthi, CeCl₃·7H2O-SiO2: catalyst promoted microwave assisted neat synthesis, antifungal and antioxidant activities of a-diaminophosphonates, Chin. Chem. Lett. 24 (2013) 759-763.

  29. [29] H. Zare, M.M. Ghanbari, M. Jamali, A. Aboodi, A novel and efficient strategy for the synthesis of various carbamates using carbamoyl chlorides under solvent-free and grinding conditions using microwave irradiation, Chin. Chem. Lett. 23 (2012) 883-886.[29] H. Zare, M.M. Ghanbari, M. Jamali, A. Aboodi, A novel and efficient strategy for the synthesis of various carbamates using carbamoyl chlorides under solvent-free and grinding conditions using microwave irradiation, Chin. Chem. Lett. 23 (2012) 883-886.

  30. [30] B. Mohammadi, M. Shafieey, H. Kazemi, A. Ramazani, Pseudo four-component and regioselective synthesis of 4-amino-3,5-dicyano-6-arylphthalates using triethylamine catalyst, Chin. Chem. Lett. 24 (2013) 497-499.[30] B. Mohammadi, M. Shafieey, H. Kazemi, A. Ramazani, Pseudo four-component and regioselective synthesis of 4-amino-3,5-dicyano-6-arylphthalates using triethylamine catalyst, Chin. Chem. Lett. 24 (2013) 497-499.

•