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Citation: ZHOU Bao-Han, CAO Hong, WANG Hong-Qing, LIU Zhao-Jie. Synthesis and Biological Activity of N-Acylpyrazole derivatives[J]. Chinese Journal of Applied Chemistry, ;2005, 22(4): 391-394. shu

Synthesis and Biological Activity of N-Acylpyrazole derivatives

1.
Department of Chemistry, Central China Normal University, Wuhan 430079

Corresponding author: LIU Zhao-Jie,
Received Date: 27 June 2004
Available Online: 7 November 2004
Fund Project: 国家计划委员会攻关项目(97-563-02-05)资助课题 (97-563-02-05)

Eleven novel N-acylpyrazole derivatives were synthesized via acylation reaction of intermediate 1H-pyrazole derivatives with acyl chloride.All the compounds synthesized were identified by means of ¹H NMR,IR and MS.These compounds show certain insecticidal activity against aphid in a dosage of 250 mg/L,and exhibit certain fungicidal activity at 50 mg/L.
- pyrethroid,
- 1H-pyrazole derivative,
- synthesis,
- bioactivity
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