Citation: Tao WANG, Si Jia XUE, Hai Jian YANG. Synthesis and Biological Activity of N-[N'-(4,5,6-Trisubstitued pyrimidin-2-yl)acetylureido] Benzoic Sulfimide Derivatives[J]. Chinese Chemical Letters, ;2000, 11(7): 581-582. shu

Synthesis and Biological Activity of N-[N'-(4,5,6-Trisubstitued pyrimidin-2-yl)acetylureido] Benzoic Sulfimide Derivatives

a Department of Chemistry, Central China University, Wuhan 430079;
b Department of Chemistry, Yichun College, Yichun 336000

Received Date: 3 December 1999
Revised Date: 14 April 2000

Fund Project: This research was supported by the Fund for Natural science of Hubei Province, China, (No:98J047)

Fourteen N'-(4,5,6-Trisubstitued pyrimidin-2-yl)-2-chloroacetylureas and fourteen N-[N'-(4,5,6-trisubstitued pyrimidin-2-yl) acetylureido] benzoic sulfimide derivatives were synthesized. Among them twenty-seven are new compounds and their structures have been confirmed by ¹HNMR, IR, MS and elemental analysis. The preliminary biological tests showed that some of the target compounds have excellent inhibitory activities against barnyard grass and rape, and the others have a good regulating activity for plant growth.
- Benzoic sulfimide,
- 2-amino-pyrimidine,
- biological activity,
- synthesis
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