Citation: Qi GAO, Lin WANG, Xiao Tian LIANG. Total Synthesis of (±)-Inophyllum B[J]. Chinese Chemical Letters, ;2002, 13(8): 714-716. shu

Total Synthesis of (±)-Inophyllum B

Institute of Materia Medica, Peking Union Medical College & Chinese Academy of Medical Sciences, Beijing 100050

Received Date: 27 November 2001

Fund Project: The authors are very grateful to professor Zhi Zhong ZHAO for his helpful discussions, and thank the National Natural Science Foundation of China for financial support (No.39970868).

(±)-Inophyllum B has been synthesized for the first time by a five-step approach from phloroglucinol, including the Pechmann reaction, Friedel-Crafts acylation, cyclization, chromenylation and Luche reduction
- (±)-Inophyllum B,
- anti-HIV-1 activity
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