Citation: Jun LIN, Sheng Jiao YAN, De Shou MAO, Rong XU, Li Juan YANG, Fu Chu LIU. Synthesis of Novel Benzoylphenylurea Chitin Inhibitors from Chlorothalonil[J]. Chinese Chemical Letters, ;2003, 14(12): 1219-1222. shu

Synthesis of Novel Benzoylphenylurea Chitin Inhibitors from Chlorothalonil

Jun LIN ^1,2, ,
Sheng Jiao YAN ^1,2 ,
De Shou MAO ¹ ,
Rong XU ¹ ,
Li Juan YANG ^1,2 ,
Fu Chu LIU ¹

1.
Department of Applied Chemistry, Yunnan University, Kunming 650091;
2.
State Key Laboratory of Elemento-organic Chemistry, Nankai University, Tianjin 300071

Received Date: 22 November 2003

Fund Project: We are grateful to the financial support of the Natural Science Foundation of Yunnan Province (1999B0005M) and the Open Foundation of State Key Laboratory of Elemento-Organic Chemistry, Nankai University.

Twenty-six novel benzoylphenylurea chitin inhibitor derivatives have been synthesized in over 30~50% yield from chlorothalonil 1 via sequential fluorine exchange, aminolysis, hydrolysis, decarboxylation and acylation reactions.
- Benzoylphenylureas,
- chitin inhibitor,
- chlorothalonil
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