Citation: Chao Zhong LI, Dong Biao ZHOU, Cheng Ye YUAN. STUDIES ON ORGANOPHOSPHORUS COMPOUNDS 69.A NOVEL SYNTHESIS OF 5-SUBSTITUTED 3-(1'-DIETHOXYPHOSPHORYLALKYL)-2-ISOXAZOLINES[J]. Chinese Chemical Letters, ;1993, 4(5): 391-392. shu

STUDIES ON ORGANOPHOSPHORUS COMPOUNDS 69.A NOVEL SYNTHESIS OF 5-SUBSTITUTED 3-(1'-DIETHOXYPHOSPHORYLALKYL)-2-ISOXAZOLINES

Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, 345 LingLing Lu, Shanghai, 200032

Received Date: 2 December 1992

Fund Project: The project was supported by National Natural Science Foundation of China.

Additions of diethyl phosphite to α-nitroalkenes followed by the introduction of trimethylchlorosilane and an activated alkene, gave the corresponding title compounds via regioselective 1,3-dipolar cycloaddition in moderate yield.
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