Citation: Yong An ZHANG, Ke Zhong LIU, Deng Yuan WANG, Yu Zhu WANG, Liang Jian QU, Chang Jin ZHU. Synthesis and Biological Activity of Philanthotoxin Analogs[J]. Chinese Chemical Letters, ;2006, 17(7): 895-898. shu

Synthesis and Biological Activity of Philanthotoxin Analogs

1.
Research Institute of Forest Ecology, Environment and Protection, CAF, Beijing 100091;
2.
The College of Agronomy, Xinjiang Agricultural University, Urumqi 830052;
3.
Department of Applied Chemistry, Beijing Institute of Technology, Beijing 100081

Received Date: 12 January 2006

Fund Project: We thank the National Key Program of China (2004BA509B12) and National Natural Science Foundation of China (No. 20372009) for their financial supports.

The synthesis of four analogs of philanthotoxin is described. The preliminary bioassay showed that these compounds all had good insecticidal activities, and the compound 6a had the best killing effect.
- PhTX,
- synthesis,
- biological activity
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