Citation: Yan ZHANG, Yun Zhen JIANG, Xiao Tian LIANG. The Synthesis of 1-(4-(N-methylsulfamylmethyl)phenyl-4-ethoxycarbonyl-2-methyl-pyrrole．A New Method of Pyrrole Synthesis[J]. Chinese Chemical Letters, ;1996, 7(10): 900-901. shu

The Synthesis of 1-(4-(N-methylsulfamylmethyl)phenyl-4-ethoxycarbonyl-2-methyl-pyrrole．A New Method of Pyrrole Synthesis

Institute of Materia Medica Chinese Academy of Medical Sciences, Peking Union Medical College Beijing 100050

Received Date: 22 April 1996

Under basic conditions 4-(N-methyl-sullamylmethyl)aniline 1 reacted with ethyl 3-bromopyruvate 2 in acetone to give the title compound 5.The structure of 5 was established by MS, IR, ¹HNMR and ¹³CNMR spectra.
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