Citation: Shui Ming LU, Wen Jing XIAO, Wen Fang HUANG, Tian Jie WU. Stereoselective Synthesis and Bioactivities of New ω-Azolyalkenes[J]. Chinese Chemical Letters, ;1998, 9(11): 997-998. shu

Stereoselective Synthesis and Bioactivities of New ω-Azolyalkenes

1.
Departmeent of Chemistry, Central China Normal University, Wuhan, 430079;
2.
Institute of Organic Systhesis, Central China Normal University, Wuhan, 430079;
3.
Center of Analysis and Testing, Central China Normai University, Wuhan, 430079

Received Date: 17 February 1998

A series of new ω-azolylalkenes 3 were synthesized by N-alkylation of obromoalkenes 2 which were obtained by Witting reaction of o-hydroxyalkylphosphonium bromide with aromatic aldehydes and subsequent bromination. The structures of products were confirmed by ¹HNMR, IR, MS and elemental analysis. The preliminary bioassay indicated that some of them had high fungicidal activities.
- Stereoselective synthesis,
- ω-azolylalkenes,
- fungicidal activities
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