Citation: Wei Yuan HUANG, Yan Song LIU, LIU Long Lü. A CONVENIENT SYNTHESIS OF FLUORINE-CONTAINING QUINOLINES[J]. Chinese Chemical Letters, ;1992, 3(8): 583-584. shu

A CONVENIENT SYNTHESIS OF FLUORINE-CONTAINING QUINOLINES

Shanghai Institute of Organic Chemistry, The Chinese Academy of Sciences, 345 Lingling Lu, Shanghai 200032

Received Date: 2 April 1992

Fund Project: This work was partially supported by the National Natural Science Foundation of China.

2-Fluoroalkyl-4-hydroxy-quinolines were easily obtained from thereactions of 2-(F-alkyl) acetates with aromatic amines in the presence of Et₃N,followed by cyclization of the intermediates with PPA.
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