Citation: Yong En GUO, Bin FU, Ying Xiang LIU. Design and Synthesis of 3, 4-Dihydropyrrolo[2, 1-c][1,4]oxazin-1-one and its 7-Acyl Derivatives[J]. Chinese Chemical Letters, ;2003, 14(10): 999-1001. shu

Design and Synthesis of 3, 4-Dihydropyrrolo[2, 1-c][1,4]oxazin-1-one and its 7-Acyl Derivatives

Department of Chemistry, Peking University, Beijing 100871

Received Date: 27 August 2002

Fund Project: This work was supported by the Scientific Research Foundation for the Returned Overseas Chinese Scholars(State Education Ministry).

Starting from 1H-pyrrole, unreported 3, 4-dihydropyrrolo[2, 1-c][1, 4]oxazin-1-one 4, 7-(4-chlorobenzoyl)-3, 4-dihydropyrrolo[2, 1-c][1, 4]oxazin-l-one 5 and 7-benzoyl-3, 4-dihydro-pyrrolo [2, 1-c][1, 4]oxazin-1-one 9 were designed and synthesized. They may have antipyretic and analgesic activities.
- 3,4-Dihydro-pyrrolo[2,1-c][1,4]oxazin-1-one,
- 7-acyl derivatives,
- synthesis,
- antipyretic,
- analgesic
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