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Citation: XU Zhi-Feng, DING Ming-Wu. Synthesis and Fungicidal Activities of 2-Alkylamino-3-aryl-5-benzyl-1-imidazolin-4-ones[J]. Chinese Journal of Applied Chemistry, ;2003, 20(10): 951-954. shu

Synthesis and Fungicidal Activities of 2-Alkylamino-3-aryl-5-benzyl-1-imidazolin-4-ones

XU Zhi-Feng ^a,, ,
DING Ming-Wu ^b

1.
a Department of Chemistry, Hengyang Normal University, Hengyang 421008;
2.
b College of Chemistry, Central China Normal University, Wuhan

Corresponding author: XU Zhi-Feng,
Received Date: 31 December 2002
Available Online: 19 May 2003
Fund Project:

The carbodiimides 4,obtained by aza Wittig reaction of iminophosphorane 3 with aromatic isocyanates, were reacted with primary alkylamines to give seven title imidazolinones 6a~6g. The structures of the compounds were confirmed by elemental analysis, IR and ¹H NMR. The cyclizing reaction of imidazolinones has a certain selectivity. The bioassay tests in vitro revealed 6e showed 71% and 65% inhibitory effect on botrytis cinerea and rhizoctonia solani, respectively.
- imidazolinone derivative,
- synthesis,
- aza Wittig reaction,
- fungicidal activity
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