Citation: Niraj K. Ladani, Divyesh C. Mungra, Manish P. Patel, Ranjan G. Patel. Microwave assisted synthesis of novel Hantzsch 1,4-dihydropyridines, acridine-l,8-diones and polyhydroquinolines bearing the tetrazolo[1,5-a]quinoline moiety and their antimicrobial activity assess[J]. Chinese Chemical Letters, ;2011, 22(12): 1407-1410. doi: 10.1016/j.cclet.2011.07.009 shu

Microwave assisted synthesis of novel Hantzsch 1,4-dihydropyridines, acridine-l,8-diones and polyhydroquinolines bearing the tetrazolo[1,5-a]quinoline moiety and their antimicrobial activity assess

Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar 388120, Gujarat, India

Received Date: 25 April 2011

Fund Project: The authors are grateful to the Department of Chemistry, S P University, India for providing laboratory facilities.

Microwave assisted efficient Hantzsch reaction via four-component coupling reactions of tetrazolo[l, 5-a]quinoline-4-carbal-dehyde, dimedone/cyclohexane-l, 3-dione, ethyl/methyl acetoacetate and ammonium acetate was described as the preparation of tetrazolo[l, 5-a]quinoline based 1, 4-dihydropyridines, acridine-l, 8-diones and polyhydroquinolines. The process presented here is simple, rapid, environmentally welcoming and high yielding. All the derivatives were subjected to an in vitro antimicrobial screening against a representative panel of bacteria and fungi and results worth further investigations.
- Microwave assisted,
- Tetrazolo[1,5-a]quinoline,
- 1,4-Dihydropyridine,
- Acridine-1,8-dione,
- Polyhydroquinoline,
- Antimicrobial activity
1. [1]
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2. [2]
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3. [3]
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4. [4]
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5. [5]
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12. [12]
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13. [13]
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14. [14]
  Hong Zhang , Cui-Ping Li , Li-Li Wang , Zhuo-Da Zhou , Wen-Sen Li , Ling-Yi Kong , Ming-Hua Yang . Asperochones A and B, two antimicrobial aromatic polyketides from the endophytic fungus Aspergillus sp. MMC-2. Chinese Chemical Letters, 2024, 35(9): 109351-. doi: 10.1016/j.cclet.2023.109351
15. [15]
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16. [16]
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18. [18]
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19. [19]
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20. [20]
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